95th Canadian Chemistry Conference and Exhibition


Organic Chemistry

Sunday AM

OR1Macleod E4

The Chemistry & Biology of Natural Products, from Coast to Coast Through the Prairies

Organizer(s) - S. Pedras, R. Andersen
Chair(s) - S. Pedras, R. Andersen

08:00 00138 How Plants Make Morphine Whether We Can Teach this Trick to a Microorganism *$Facchini P.J.
08:40 00139 Natural Product Genomics: Elucidating Cannabinoid Biosynthesis in Cannabis sativa Page J.E.
09:20 00140 Biosynthetic Puzzles: The Cruciferous Phytoalexins Rapalexin A and Isocyalexin A Yaya E.E., $Pedras M.S.C.
09:40 00141 meso-2,3-Butanediol: A Bacterial Metabolite with Possible Implications in Bowel Disease *$White R.L., Resmer K.L., Moussa N.T.
10:00 Coffee Break
10:20 00142 Assembly of Bioactive Macrolides by Fungal Polyketide Synthases *$Vederas J.C.
11:00 00143 Natural Product Biosynthesis in Northern Manitoba Lichen and Other Fungi Piercey-Normore M., Abdel-Hameed M., Weessies C., Anyanwu C.S., Nadeau A.K., *$Sorensen J.L.
11:20 00144 The Biosynthesis of b-Lactones *$Harrison P.H.M., Ahilan Y.
12:00 00145 Modulation of Starch Digestion for Slow Glucose Release Through "Toggling" of Activities of Mucosal a-Glucosidases $Pinto B.M.
12:20 End of Session

OR2Macleod C

Symposium on Homogeneous and Heterogeneous Catalysis in Honour of Howard Alper (joint with IN)

Organizer(s) - C. Crudden
Chair(s) - C. Crudden

08:00 00146 Abiological Self-Assembly: Predesigned Metallacycles and Metallacages via Coordination *$Stang P.J.
08:40 00147 Discovery of Sustainable Catalytic Reactions Based on Metal-Ligand Cooperation Milstein D.
09:20 00148 Mechanistic Studies in the Service of Asymmetric Gold(I) Catalysis Gagne M.
10:00 Coffee Break
10:20 00149 Enantioselective Photoredox Organocatalysis: A New Catalysis Concept of Broad Utility to Chemical Synthesis *MacMillan D.W.C.
11:00 00150 Kinetic Profiling as a Tool for Illuminating Important Off-Cycle Catalyst Reservoirs in Organocatalytic Reactions *$Hein J.E.
11:20 00151 Metal Free Catalytic Hydroborations Bailey A.M., *Eisenberger P., $Crudden C.
11:40 00152 Organocatalytic Asymmetric Conjugate Additions of Heteroaryl Moieties to a,b-unsaturated Enones with Boronates and 3,3³-Disubstituted Binaphthols Cheung D.C.Y., $Chong J.M.
12:00 00153 Nickel Perfluorometallacycles: Intermediates for Sustainable Routes to Functionalized Fluorocarbons? Giffin K.G., *Harrison D.H., $Baker T.B.
12:20 End of Session

OR5Macleod B

Small Molecule Drug Design and Development

Organizer(s) - J. Wulff
Chair(s) - J. Wulff, S. Chowdhury

08:40 00154 Timely Chemical Process Research is a Critical Part for Efficient Drug Development Senanayake C.
09:20 00155 Disrupting the Histone Code: Inhibition of Histone-Reader Protein Interactions as a Novel Approach to Cancer Therapeutics *$Hof F., Daze K.D., Pinter T., Ma M.C.F., Pineux F.
09:40 00156 Bestowing Peptides with Small Molecule Properties Zaretsky S., Scully C., Ler S., Yu J., $Yudin A.K.
10:00 Coffee Break
10:20 00157 Design and Synthesis of Novel Antimicrobials based on a Putative Endogenous Antibacterial Wu F., Henneberry A., Lu E., Barden C., Byers D., McMaster C., *$Weaver D.
11:00 00158 Synthesis of a Unique 7a-Testosterone-chlorambucil Hybrid Showing Selectivity on Hormone-dependent Prostate Cancer Cells *$Bérubé G., Bastien D., Hanna R., Leblanc V., Asselin É.
11:20 00159 Structure-Activity Relationship of Imidazolium-based Synthetic Anion Transporters *Elie C.R., Charbonneau M., $Schmitzer A.R.
11:40 00160 Metabolic Optimization of Potent Stat3 Inhibitors for Improved Cancer Therapeutic Agents *Arpin C.C., Page B.D.G., Turkson J., $Gunning P.T.
12:00 00161 Semi-Synthesis of a Biologically Inspired Library of Natural Product Mimics from Lypophillic Marine Natural Product b-gorgonene Pearce B., $Kerr R., *McCulloch M.
12:20 End of Session

OR6TELUS 106

Applied Photochemistry in Health Research (joint with BM)

Organizer(s) - B. Heyne
Chair(s) - S. Mooi

08:40 00162 Fluorogenic Protein Labelling *$Keillor J.W., Pardin C., Strmiskova M., Chen Y.
09:20 00163 Quantitative Synthesis of Genetically Encoded Libraries of Light-responsive Ligands Jafari M.R., Ng S, *$Derda R
09:40 00164 Towards a Fluorometric Assay for Human Factor XIIIa Mulani A., $Keillor J.W., Cormier M., Poirier M.
10:00 Coffee Break
10:20 00165 Development of Small Latent Fluorophore Substrates for the ATG4B Enzyme Vezenkov L.L., Kumar N.S., Nguyen T.G., *$Young R.N.
10:40 00166 Novel Quantum Yield Modulation Mechanism of an RFP-based Ca2+ Biosensor Carlson H.J., $Campbell R.E.
11:00 00167 Computationally Guided Engineering of Conformationally Flexible Green Fluorescent Protein Abdelfattah A.S., *$Campbell R.E.
11:20 00168 Fluorescence Visualization, from Reactive Oxygen Species in Cell Membranes to Biomolecular Structures at the Single Molecule Level *$Cosa G.
12:00 End of Session

ORMacleod E1

Ligand Design (joint with IN4)

08:00 See IN4.

12:20 End of Session

ORGlen 202

Modern Methods in Polymer Synthesis (joint with MS4)

08:40 See MS4.

12:20 End of Session

ORMacleod D

Molecular Design of Optical, Photonic and Electronic Materials

08:00 Joint with MT and IN - See MT2.

12:20 End of Session


Sunday PM

OR1Macleod E4

The Chemistry & Biology of Natural Products, from Coast to Coast Through the Prairies

Organizer(s) - S. Pedras, R. Andersen
Chair(s) - S. Pedras, P.H.M. Harrison

13:40 00502 Natural Product Discovery from a Marine Microbial Library Kerr R.
14:20 00503 Characterizing Myxobacterial Polyketide Biosynthetic Pathways from Whole Genome Sequencing *$Boddy C.N., Conway K., Taylor R.E., Young J.
15:00 00504 Anti-Mycobacterial Natural Products from Canadian Traditionally Used Medicinal Plants and their Endophytic Fungi *$Gray C.A., Johnson J.A., Webster D.
15:40 Coffee Break
16:00 00505 Biosynthesis of Ethyl Oleate in Honey Bees *$Plettner E., Castillo C., Chen H.
16:40 00506 The UVA and Aqueous Stability of Flavonols Under Investigation as Topical Skin Photoprotectants Maini S., Hodgson H.L., *$Krol E.S.
17:00 00507 Expression and Analysis of Cryptic Biosynthetic Genes in Streptomyces Kalan L., Gessner A., Bechthold A., Wright G.D., *$Zechel D.L.
17:20 End of Session

OR2Macleod C

Symposium on Homogeneous and Heterogeneous Catalysis in Honour of Howard Alper (joint with IN)

Organizer(s) - C. Crudden
Chair(s) - C. Crudden

13:40 00508 Catalytic Use of Carbon Monoxide in Synthesis Murai S.
14:00 00509 Ni Catalyzed C-F Activation: New Methods for the Synthesis of Novel Aryl Fluoride Building Blocks Keyes L., *Yeo C.F.H., $Love J.A.
14:20 00510 Synthesis of Acetylenes by Combination of Sonogashira Coupling and Double Elimination Protocol of b-Substituted Sulfone *Orita A., Yang X., Xu F., Peng L., Suzuma Y., Otera J.
15:00 00511 Multi-Component Coupling Processes by Pd/Light Accelerated Atom Transfer Carbonylation of Alkyl Iodides Ryu I.
15:40 Coffee Break
16:00 00512 New Catalysts for Carbonylation and Carboxylation *$Nozaki K.
16:40 00513 A Practical Mechanistic Update on the Copper-Catalyzed Azide-Alkyne Click Reaction *$Finn M., Rodionov V.O., Hong V.P., Presolski S.I.
17:20 End of Session

OR5Macleod B

Small Molecule Drug Design and Development

Organizer(s) - J. Wulff
Chair(s) - P. Forgione, A. Scholte

13:40 00514 Design and Synthesis of Novel Drugs for the Treatment of Heart Failure and Cardiac Arrhythmias *Back T.G., Smith C.D., Wang A., Vembaiyan K., Chen S.R.W.
14:00 00515 Glutamate-1-semialdehyde Aminomutase Inhibitors as Potential New Antibiotics Patel T., Taj R., Nadeau A.K., Stetefeld J., *$Sorensen J.L.
14:20 00516 Identification of Novel Androgen Receptor Antagonists by Molecular Design Wu J.H.
15:00 00517 Tetrapodal Salicylic Acid-based Inhibitors of Stat3 Protein Demonstrate Potent Activity Against Multiple Myeloma in Pre-clinical studies Page B.D.G., Li Z.H., Atkninson J., Wong Y.L., Haftchenary S., Croucher D.C., Jimenez-Zepeda V.H., Spagnuolo P.A., Turkson J., Schimmer A.D., Trudel S., *$Gunning P.T.
15:20 00518 Synthesis and Properties of Molecular Probes for Cystic Fibrosis Research Alkhouri B., *$Viirre R.D.
15:40 Coffee Break
16:00 00519 Prevention of Intestinal Iron Uptake by Inhibition of Human Divalent Metal Transporter 1 (DMT1) With A Novel Small Molecule Inhibitor, XEN601 *Chowdhury S., Cadieux J., Chahal N., Fu J.-M., Grimwood M., Huang J., Zhang Z., Brownlie-Cutts A., Mattice M., Lin S., Webb M., Ratkay L., Waldbrook M., Xie C., Samra P., Sojo L., Mansour T., Goldberg P.Y., Hayden M., Pimstone S., Cohen C.
16:20 00520 Development of a Drug Screening Assay for b-Amyloid Antiaggregants Meier-Stephenson F.S., Fisher L.K., McGrath A.J., *$Weaver D.F.
16:40 00521 Salicylic Acid Mimetics and Prodrugs Targeting Transcriptionally Active STAT3 in Brain Cancer Cells Haftchenary S., Luchman A., Dawson S., Page B.D.G., Shahani V.M.S., Weiss S., Turkson J., $Gunning P.T.
17:00 End of Session

OR6TELUS 106

Applied Photochemistry in Health Research (joint with BM)

Organizer(s) - B. Heyne
Chair(s) - B. Heyne

13:40 00522 Control of the Speed for Guest Release from Supramolecular Systems. Insights from Studies on the Dynamics of Host-guest Complexes *$Bohne C.
14:20 00523 Synthesis of Photochromic Asymmetrical Dithienylethene Derivatives Kandasamy Y., *$Murphy R.S.
14:40 00524 Photoisomerization at High External Pressures: Testing the Strength of a Light-activated Molecular Muscle Singleton T.A., Ramsay K.S., Barsan M.M., Butler I.S., *$Barrett C.J.
15:00 00525 Photobleaching Kinetics of Verteporfin and Lemuteporfin in Cells and Optically Trapped Multilamellar Vesicles Using Two-photon Excitation Tekrony A.D., Kelly N.M., Fage B.A., $Cramb D.T.
15:20 00526 The Unexpected Photochemistry of a 7-Nitrobenzofurazan Derivative Sveen C., Zaremberg V., *$Heyne B.
15:40 Coffee Break
16:00 00527 A New Way to View Organization - Size Matters Mooi S., $Heyne B.
16:20 00528 Using Lanthanide-Doped Upconverting Nanoparticles for the "Remote-Control" of Photochemical Reactions Boyer J.-C., Carling C.-J., *$Branda N.R.
16:40 00529 Photothermal Effect of Silicon Nanocrystals Regli S., Kelly J.A., Shukaliak A.M., *$Veinot J.G.C.
17:00 End of Session

OR8Macleod A1

General

Organizer(s) - T. Sutherland
Chair(s) - S. Keller

13:40 00530 A Turn-On Fluorogenic Probe for MDMA from Ecstasy Tablets Moreno D., Diaz de Grenu B., Garcia B., Ibeas S., *$Torroba T.
14:00 00531 Calixarene-derived Aromatic Cages for Binding Biologically Importantant Cations in Water Whiting A.L., Daze K.D., Ma M.C.F., Dubicki K.I., *$Hof F.
14:20 00532 Exploring Tetrazoles and Other Carboxylic Acid Bioisosteres as Novel Agents for Anion Binding, Sensing and Transport Pinter T., $Hof F.
14:40 00533 Cyclodextrin Derivatives with Liquid Crystal Properties Ward S., $Ling C.C.
15:00 00534 Cucurbituril Host-Guest Complexes with Acridizinium Cations Fraser A.J., *$Macartney D.H.
15:20 00535 Cucurbituril Complexes of Steroidal Neuromuscular Blocking Agents Gamal-Eldin M., *$Macartney D.H.
15:40 Coffee Break
16:00 00536 5-Exo-dig Cyclizations Toward Isoindolinone-Containing Oligomers, Macrocycles, and Molecular Switches *$Eisler S., Bubar A., Estey P., Lawson M.
16:20 00537 Synthetic Cationic Lipids *Parvizi P., $Fyles T.M.
16:40 00538 Synthesis, Characterization and Properties of a New Pyrene-Based BINOL Derivative MacKinnon M.R., *Bodwell G.J.
17:00 00539 Chiral BINOL-imidazolium Salts and their Applications in Catalysis Vidal M., $Schmitzer A.R.
17:20 End of Session

ORMacleod E1

Ligand Design (joint with IN4)

13:40 See IN4.

17:20 End of Session

ORGlen 202

Modern Methods in Polymer Synthesis (joint with MS4)

13:40 See MS4.

16:40 End of Session

ORMacleod D

Molecular Design of Optical, Photonic and Electronic Materials

13:40 Joint with MT and IN - See MT2.

17:40 End of Session


Monday AM

OR1Macleod E4

The Chemistry & Biology of Natural Products, from Coast to Coast Through the Prairies

Organizer(s) - S. Pedras, R. Andersen
Chair(s) - S. Pedras, E. Plettner

08:00 00689 Applications of Phytohormone Signaling Manipulation Towards Crop Improvement *Abrams S.R., $Nelson K.M., Zaharia L.I.
08:40 00690 Plant Natural Products with Enzyme Inhibitory Activities *$Ata A.
09:20 00691 Cladoniamide Biosynthetic Gene Cluster *Ryan K.S., Du Y.-L.
10:00 Coffee Break
10:20 00692 Structural Diversification, Biosynthetic Insights and Mechanism of Action Studies on the Jadomycins *$Jakeman D.L.
11:00 00693 New Tools for the Characterization of Natural Products *$Derksen D.J.
11:20 00694 Computational and Electrophysiological Studies of (+)-Disparlure Analogs with Gypsy Moth Pheromone Binding Proteins Yu Y., $Plettner E.
11:40 00695 Metabolomic Mining of Microbiomes for Bioactive Natural Products Ibrahim A., Yang L., Ma B., Magarvey N., Cheriton D.
12:20 End of Session

OR2Macleod C

Symposium on Homogeneous and Heterogeneous Catalysis in Honour of Howard Alper (joint with IN)

Organizer(s) - C. Crudden
Chair(s) - C. Crudden

08:00 00696 Mixed-valent, Phosphoranimide-supported First-row Metal Clusters for Catalytic Deep Hydrodesulfurization Under Mild Conditions Brown H.J.S., $Stryker J.M., Ferguson M.J.
08:20 00697 The Catalytic Reduction of Ketones and Imines Using Iron-based Precatalysts : Catalysis and Mechanistic Insight Mikhailine A.A., *Maishan M.I., $Morris R.H.
08:40 00698 Chlorometallate Ionic Liquids Revisited Estager J., Seddon K.R., Swad'ba-Kwa'ny M.
09:20 00699 Phosphonium Ionic Liquids as Ruthenium Nanoparticle Stabilizers and Ligands to Rhodium Complexes: Applications to Catalysis of Hydrogenation and Hydroformylation Luska K.L., Demmans K.Z., Stratton S.A., *$Moores A.
09:40 00700 Amphoteric a-Boryl Aldehydes and their Use in Generating Complex Building Blocks via a-Functionalization St. Denis J.D., *$Yudin A.K.
10:00 Coffee Break
10:20 00701 STEM Education in American Public Research Universities *$Fox M.A.
11:00 00702 Cross-Coupling Reactions Have Enhanced Functional Elemento-Organic Chemistry Tamao K.
11:40 00703 Phosphino - Imidazoline Ligands in Homogeneous and Polymer-supported Catalytic Systems *Claver C., de la Fuente V., Castillon S., Marcos R., Couso X., Pericas M.
12:20 End of Session

OR5Macleod B

Small Molecule Drug Design and Development

Organizer(s) - J. Wulff
Chair(s) - A. Scholte, J. Wulff

08:40 00704 The Resurgence of Covalent Drugs *Petter R.C.
09:20 00705 Development of Novel Hybrid VDR Agonist / HDAC Inhibitors for Cancer Treatment *$Gleason J.L., White J.H., Fischer J., Wang T.T., Kaldre D., Moras D., Rochel N.
09:40 00706 Development of a New Class of Neuraminidase Inhibitors for the Treatment of Oseltamivir-Resistant Influenza and Other Circulating Influenza Strains Brant M.G., Mason J.W., *Bromba C.M., $Wulff J.E.
10:00 Coffee Break
10:20 00707 Progress Toward a STAT3 Small Molecule Therapeutic for the Treatment of Breast and Brain Cancers *$Gunning P.T.
11:00 00708 3-Hydroxyanthranilate Antiaggregants: NMR-Based Explorations of Non-Covalent Binding to Amyloid-Beta *Weaver D.F., Meek A., $Simms G.A.
11:20 00709 Synthesis of Novel Sym-Triazine Compounds as Multi-Target-Directed Ligands for Alzheimer's Disease Dhar D., Mikhaylichenko S., Veloso A.J., $Kerman K.
11:40 00710 Synthesis of New Benzopyrano Imidazole Derivatives for Antihypertensive Activity *$Ghate D.M., Bano M., Ivanov I.
12:00 00711 Disulfide-bridged Peptide Macrocycles: Versatile Tools for Microarray Applications Chung B.K.W., *Hickey J.L., $Yudin A.K.
12:20 End of Session

ORMacleod E1

Ligand Design (joint with IN4)

08:00 See IN4.

12:20 End of Session

ORMacleod D

Molecular Design of Optical, Photonic and Electronic Materials

08:00 Joint with MT and IN - See MT2.

12:20 End of Session

ORTELUS 105

Teaching Organic Chemistry (joint with CE3)

10:20 See CE3.

12:20 End of Session


Monday PM

OR2Macleod C

Symposium on Homogeneous and Heterogeneous Catalysis in Honour of Howard Alper (joint with IN)

Organizer(s) - C. Crudden
Chair(s) - C. Crudden

13:40 00959 Z-selective Ruthenium-based Catalysts for Olefin Metathesis Occhipinti G., Hansen F.R., *Jensen V.R.
14:00 00960 Chemical Plants? Olefin Metathesis as a Tool for Capturing Naturally-Occurring, High-Value Structural Motifs Lummiss J.A.M, dos Santos E.N., Oliveira K.C., *$Fogg D.E.
14:40 00961 Mechanistic and Developmental Catalytic Hydrogenations of Amides, Imides, and Ketones *$Bergens S.H., John J.M., Takebayashi S.

Canadian Council of University Chemistry Chairs (CCUCC) Chemistry Doctoral Award lecture:

15:00 00962 Transition Metal Catalysis: Activating CO2, CH, and CO Bonds En Route to Carboxylic Acids, Biaryls, and N-Containing Heterocycles Yeung C.S., *Dong V.M.
15:40 Coffee Break
16:00 00963 A Rhodium Catalyst-Organic Framework for the Intramolecular Cycloisomerization of 1,6-Enynes Corkum E.G., Hass M.J., Sullivan A.D., *$Bergens S.H.
16:20 00964 The Selective Oligomerisation of Ethylene to 1-Hexene and 1-Octene Green M.
17:00 00965 Pd- or Ni-Catalyzed Addition of R2P(O)-E (E = H, SR') with Alkynes *$Tanaka M.
17:40 End of Session

OR8Macleod E4

General

Organizer(s) - T. Sutherland
Chair(s) - T. Sutherland

13:40 00966 Induction of Metabolic Variations in the Fungal Pathogen Alternaria brassicicola Park M.R., $Pedras M.S.C.
14:00 00967 Metabolism of Camalexins and Analogs by the Cruciferous Pathogen Alternaria brassicicola Abdoli A., $Pedras M.S.C.
14:20 00968 Synthesis of Amanitin and Bioactive Derivatives of Trypathionine-containing Peptide Natural Products *$Perrin D.M., Zhao L., Blanc A., Dietrich D.J.
14:40 00969 Total Synthesis of Vallartanone A: Strategic Coupling of Chiral Fragments via Kinetic Resolution Lai L.C. K., $Ward D.E.
15:00 00970 Dhilirolides A-N, Meroterpenoids Produced in Culture by the Fruit-Infecting Fungus Penicillium purpurogenum Collected in Sri Lanka de Silva E.D., Williams D.E., Jayanetti D.R., Centko R.M., Patrick B.O., Wijesundera R.L.C., Andersen R.J.
15:20 00971 Toward Mechanistic Studies of Cyclopropane Desaturases: Enantioselective Synthesis of (9S,10R)-Dihydrosterculic Acid Palko J.W., Buist P.H., *$Manthorpe J.M.
15:40 Coffee Break
16:00 00972 Isolating and Studying Hyperconjugation with the Conformational Isotope Effect: an Experimental and Theoretical Study Greenway K.T., Bischoff A.L., *$Pinto B.M.
16:20 00973 Thermodynamics of Lewis Acid-Base Complexation of Transient Silylenes and Germylenes with Chalcogen and Pnictogen Donors by Laser Flash Photolysis Techniques Kostina S.S., *$Leigh W.J., Singh T.
16:40 00974 The Direct Detection and Characterization of Transient Stannylenes in Solution by Laser Flash Photolysis Methods Duffy I.R, *$Leigh W.J.
17:00 End of Session

OR-PoExhibition Hall CD

Poster Session

From 18:00 until 19:30

18:00 00975 Rewards and Profit from Applied Organic Syntheses *$Lynch B.M., Ceretti E.
18:00 00976 Preparation and Characterization of New Organosoluble Polyamides with Good Thermal Properties Containing Photosensitive Group in the Main Chain *$Hajibeygi M., Shabanian M.
18:00 00977 Design, Synthesis and In Vitro Evaluation of Arginine and Citrulline Modified PARACEST MRI Contrast Agents: Can the Nitric Oxide Synthase (NOS) Enzymatic Activity be Detected by MRI? Suchy M., Li A.X., Milne M., Bartha R., Hudson R.H.E.
18:00 00978 b-Arylation of Aldehydes Pirnot M.T., Rankic D.A., Martin D.B.C., *$MacMillan D.W.C.
18:00 00979 Absolute Configuration and Predominant Conformations of a Chiral Crown Ether-based Colormetric Sensor: A Vibrational Circular Dichroism Spectroscopy and DFT Study of Chiral Recognition Merten C., Hyun M.H., *Xu Y.
18:00 00980 Mild and Convenient Synthesis of 1,2,3 - Triiodoarenes and Their Applications in One-Pot Tandem Reaction *$Al-Zoubi R.M., AbulFutouh H.
18:00 00981 Novel and Efficient Synthesis of Tetrazolo[1,5-b]-1,2,5-Oxadiazepines and Assessment of their Antibacterial Activities El-Badry S.M., *$Taha M.A.
18:00 00982 An aza-Wittig Approach to Sulfinimines and Sulfonamides from Sulfonyl Azides McConkey C., Ratiani M., $Hill B.
18:00 00983 Synthesis of 3-Substituted 3-Arylpropanols by the Truce-Smiles Rearrangement Grewal R., Kosowan J., W'Giorgis Z., *$Wood T.E.
18:00 00984 Towards the Total Synthesis of Palmyrolide A *Hood M., $Magee D.I.
18:00 00985 Dianthryl-TTFV as Dual Functional Fluorescent Probe for Transition Metal ions and Specific Anions Mulla K., Dongare P., Thompson D.W., *Zhao Y.
18:00 00986 Diazapolyenes and Borylated Azapolyenes: Synthesis of Nitrogen/Boron-Containing Heterocycles and their Properties Neue B., Fröhlich R., *Würthwein E.-U., Wakamiya A., Fukazawa A., Yamaguchi S.
18:00 00987 On the Origin of Stereocontrol in Enantioselective Diels-Alder Reactions from Aldehydes Mak C.C., *$Muchall H.M.
18:00 00988 Synthesis and Self-Assembly of New guanine-cytosine Motifs $Legesse B., Oderinde M., *Fenniri H.
18:00 00989 Brassinosteroids: New Synthetic Strategy and Neuroprotective Activity Ismaili J., Martinoli M.-G., Longpré F., $Daoust B.
18:00 00990 Cleavage of DNA using Two-Photon Excitation of N-Alkoxypyridinethiones Ruzic-Gauthier M., Cozens F.L., *$Schepp N.P.
18:00 00991 Synthetic Studies Towards Palau'amine: Synthesis of trans-fused 5,5-ring Systems and Advances in an Oxidative Cyclization Sequence Rivalti D., $Gleason J.L.
18:00 00992 Synthesis of 5- and 6-Membered Cyclic Hydrazides as Organocatalysts for Cycloaddition Reactions Biggs R.A., $Ogilvie W.W.
18:00 00993 Cascading Radical Cyclization of Bis-vinyl Ethers: A Mechanistic Investigation $O'Rourke N.F., Davies K.A., *Wulff J.E.
18:00 00994 An Approach Toward the Total Synthesis of Didemnaketal A $Davy J., Bromba C., Moreau B., *Wulff J.
18:00 00995 Synthetic Substrates for a New Capillary Electrophoresis Laser-Induced Fluorescence Protease Activity Assay Wiebe M., Craig D.B., *$Wood T.E.
18:00 00996 Synthesis of Hydroxamic Acid Histone Deacetylase-6 Inhibitors and Evaluation of Isoform Selectivity W'Giorgis Z., *$Wood T.E.
18:00 00997 Tripeptide Chymotrypsin Substrates for a New Capillary Electrophoresis Laser-Induced Fluorescence Activity Assay Kosowan J., Craig D.B., *$Wood T.E.
18:00 00998 Investigation of Substituent Effects Upon the Truce-Smiles Rearrangement of Nitrophenoxy 3-Butyronitrile Aryl Ethers Grewal R., *$Wood T.E.
18:00 00999 Effect of Zeolite Composition on Two-Photon Absorption of Simple Organic Chromophores Pettipas S., Cozens F.L., *$Schepp N.P.
18:00 01000 Supramolecular Assistance In Assymetric Catalysis Gravel J., Gauchot V., *Schmitzer A.R.
18:00 01001 High Pressures to Promote Diels-Alder Reactions Between Diazo Compounds and Various Dienes Landschoot B.K., *Humenny W.J., $Kerr M.A.
18:00 01002 Useful Molecular Complexity Generated by a Gramine-type Fragmentation of a Meldrums Acid Moiety Armstrong E.L., $Kerr M.A.
18:00 01003 Towards the Synthesis of a New Pd-Phosphine Catalyst for the Buchwald-Hartwig Reaction Chojnacka M.W., Viirre R.D., Gossage R.A.
18:00 01004 Synthesis and Investigation of the Liquid Crystalline Properties of Novel Substituted Dibenzanthracenes Psutka K.M., Williams J., Paquette J., *$Maly K.E.
18:00 01005 meso-Functionalized BODIPY Dyes: Effect of C2 and C6 Substitution on Electrophilicity, Photostability and Excited State Energy Levels Lincoln R., Greene L., Krumova K., $Cosa G.

OR1 - The Chemistry and Biology of Natural Products posters

18:00 01006 Phytochemical Analysis of Boreal Draba (Draba borealis DC, Brassicaceae) *$Montaut S., Chiari L., Montagut-Romans A.
18:00 01007 Mechanistic Investigations of DcsC, a PLP-independent Racemase Dietrich D., van Belkum M.J., *$Vederas J.C.
18:00 01008 Chemistry of Haircolor: Advantages and Disadavantages *$Nazari M., Nazari K.
18:00 01009 Anti-Renin Alkaloids from Nauclea latifolia Agmouh A.A., Sintra E.R., *$Ata A., Aluko R.E.
18:00 01010 Phytochemical Studies on Genus Buxus Lam C.W., Al-Malki M., Gengan R.M., *$Ata A.
18:00 01011 Sequencing the Putative Usnic Acid Polyketide Synthase Gene *Abdel-Hameed M., $Sorensen J.
18:00 01012 The Ring-Closing Metathesis of Unprotected Peptides in Water Cochrane S.A., Huang Z., *$Vederas J.C.
18:00 01013 Incorporation of Partially Assembled Intermediates by the Hypothemycin Polyketide Synthase Norquay A.K., Gao Z., *Vederas J.C.
18:00 01014 A Fungal Ketoreductase Domain that Displays Substrate-dependent Stereospecificity Gao Z., *$Vederas J.C.
18:00 01015 Preparation of Fluorescent Analogues of Neopetrosiamide Towle K.M., Chaytor J.L., Liu H., *$Vederas J.C.
18:00 01016 Synthesis of Phosphopantetheine Thioesters to Investigate the Function of the Condensation Domain in the Biosynthesis of Lovastatin Cochrane R.V.K., Chaytor J.L., Hawranik D.J., *$Vederas J.C.
18:00 01017 Active Site Studies of Arogenate Dehydrogenase & the Purification of its Substrate Rachel N., $Turnbull J.L.
18:00 01018 Synthesis of Phosphonates to Characterize Enzyme-Substrate Interactions in Macrolactonization Argyropoulos P., Pinto A., *$Boddy C.N.
18:00 01019 Progress Toward the Total Synthesis of Scandine and the Melodinus Alkaloids Goldberg A.F.G., Stoltz B.M.

OR2 - Symposium on Homogeneous and Heterogeneous Catalysis in Honour of Howard Alper posters

18:00 01020 Study of 9-anthraldehyde Oxidation with Surface Plasmon Band Irratdiation of Photochemical Synthethized Diamond Supported Gold Nanoparticles *Wee T.L., Schmidt L.C., $Scaiano J.C.
18:00 01021 New Chiral Ligands From 2,5-anhydro-D-mannitol: Towards the Application in Asymmetric Transfer Hydrogenation Soueidan O.M., Kondapi V., *West F.G.
18:00 01022 Toward Efficient and Green Nanobiocatalysis by the Nanostructured Porous Materials $Salehi Siavashani E., *Adhami F., Nazari K.
18:00 01023 Catalysis with Boron Eisenberger P., Bailey A.M., $Crudden C.M.
18:00 01024 Hydrogenation of Disubstituted Arenes with Metal Nanoparticles as Catalysts *Claver C., Godard C., Llop J.
18:00 01025 Phosphorus-Containing Copolymers for Supported Catalysis Hey T.W., Hsieh T., $Gates D.P.
18:00 01026 Syntheses of Fluoroalkyltin Clusters and Their Applications to Carbon-Carbon Bond Forming Reactions *Orita A., Tokunaga T., Otera J.
18:00 01027 Nanoparticle Catalyzed Redox Processes in Tetraalkylphosphonium Ionic Liquids Banerjee A., $Scott R.W.J.
18:00 01028 Chemoselectivity of the Suzuki-Miyaura Reaction with Aryl Secondary Boronic Esters Moore B., $Crudden C.M.
18:00 01029 Mono(2-Aminopyridinato) Titanium Catalyst for Aminoalkene Hydroamination Chong E., $Schafer L.L., Kempe R.
18:00 01030 Synthesis and Nucleophilic Reactivity of Cobalt Fluorocarbenes Harrison D.J., Lee G.M., Gorelsky S., Korobkov I., *$Baker R.T.
18:00 01031 Asymmetric Homogeneous Hydrogenation of Unsaturated Carboxylic Acids de Winter T., *$Jessop P.
18:00 01032 Selective a-Alkylation of Saturated N-Heterocycles via Hydroaminoalkylation using Tantalum Amidate Precatalysts Payne P.R., *Eisenberger P., $Schafer L.L.
18:00 01033 Solvent-Free Isomerizations of Allylic Alcohols Catalyzed by a Rhodium Catalyst-Organic Framework Corkum E.G., Kalapugama S., Hass M.J., *$Bergens S.H.
18:00 01034 Ruthenium Catalyzed Asymmetric Hydrogenation of Racemic a-Chiral Amides: Accessing Amines and Chiral Alcohols Via Dynamic Kinetic Resolution John J.M., *$Bergens S.H.
18:00 01035 The Suzuki Reaction: a Mechanistic and Kinetic Study by ESI-MS Logan J.R., *McIndoe J.S., Ahmadi Z.

OR3 - Symposium in Honour of Edward Piers posters

18:00 01036 Aziridine-2-carboxylic Acid-containing Cyclic Tetrapeptides: Synthesis and Reactivity White C.J., $Yudin A.K.

OR4 - Advances in Synthetic Methods posters

18:00 01037 Pronounced Ligand Effects in the First Well-defined Silver(I)-Complex-Catalyzed Cycloaddition of Azides onto Terminal Alkynes Keskar K., *$McNulty J.
18:00 01038 Development of New Methodologies for the Construction of C-C and C-N Bonds Using Alkylbismuth Reagents *$Gagnon A.
18:00 01039 The Total Synthesis of (R)-8-hydroxy-6,7-dimethoxy-1-(4-iodobenzyl)-2-((R)-1-phenylethyl)-1,2,3,4-tetrahydroiso- quinoline (1) the Precursor of Bisbenzyltetrahydroisoquinoline Alkaloids (-)-cycleanine Dakhil O., *Georghiou P.
18:00 01040 Electrophile-Induced Rearrangement Reactions of Vinylboronates for C-C Bond Formation Yakiwchuk J., Fainman S., *$McCubbin J.A.
18:00 01041 Allylic Alcohol Rearrangement - Diels-Alder Sequence for the Synthesis of Bi- and Tricyclic Ring Systems Voth S., *$McCubbin J.A.
18:00 01042 Formation of Optically Pure Cyclic Amines by Intramolecular Conjugate Displacement Cheng P., Clive D.L.J.
18:00 01043 Efforts Towards an Asymmetric Suzuki-Miyaura Cross-Coupling of Polyboronylalkanes with Aryl Halides Sun H.-Y., *$Hall D.G.
18:00 01044 Stereoselective Installation of Carbon-Heteroatom Bonds Using Amphoteric Molecules Liew S.K., $Yudin A.K.
18:00 01045 SNAr and Nitrile Hydrolysis using KF/Alumina Under Solvent-free Conditions Jones-Mensah E., Durrant J., *$Magolan J.
18:00 01046 Novel Lewis Acid Promoted Asymmetric Diels Alder Reactions Warner T.G., $Keay B.A.
18:00 01047 A Dieckmann Cyclization Route to 2,5-Piperazinediones *Larrivee Aboussafy C., $Clive D.L.J.
18:00 01048 Mild Vanadium Catalyzed Desymmetrization of Tertiary Allylic Alcohols Fradette R.J., Rieder C.J., *$West F.G.
18:00 01049 A Novel Approach Towards the Synthesis of Faveline- and Icetexane-Diterpenes by Electrophilic Cyclization of Vinylogous Propargyl-Acetate-Co2(CO)6 Complexes Kolodziej I., $Green J.R.
18:00 01050 Solvent-free Aerobic Dehydrogenation on the Surface of Ferric Oxide and Silica Karki M., Araujo H., *$Magolan J.
18:00 01051 An Efficient One-Pot Synthesis for 1,2-disubstituted Tetrazoles from Amide Precursors Maillet R., $Ling C.C.
18:00 01052 An Approach Towards the Enantioselective Construction of the Tetracyclic Core of the Sarpagine Alkaloids Hughes J.M.E., *Wee A.G.H.
18:00 01053 Synthesis of Heteroaromatics via One-pot Solvent-free Cyclization and Aerobic Dehydrogenation Araujo H., Karki M., *$Magolan J.
18:00 01054 Efficient Synthesis of Benzimidazoles using Two Heterogeneous Catalysts in One Pot Weires N.A., Boster J., *$Magolan J.

OR5 - Small Molecule Drug Design and Development posters

18:00 01055 Boron-Containing Capsaicin Derivatives for the Treatment of Cancer Ramsaywack S., Decken A., Fontaine F.-G., Culf A.S., *$Westcott S.A.
18:00 01056 Synthesis and Cytocidal Activity of a Series of 7a-Testosterone Amides as Potential Anticancer Agents *$Bérubé G., Morin N., Bruneau J., Brasseur K., Leblanc V., Asselin É.
18:00 01057 Development of Novel anti-Influenza Virus A Agents Adabala P.J., Mohan S., *$Pinto B.M.
18:00 01058 Thieno[2,3-d]pyrimidinone Derivatives as Small Molecule Inhibitors of the Prevalent Pseudomonas aeruginosa Virulence Factor Exotoxin A in Patients with Cystic Fibrosis *Shkoor M., Rochon A., $Schwan A.
18:00 01059 Synergistic Modulation of Stereochemistry and Side-chain-to-backbone Cyclization in Anti-inflammatory Peptide Mimic Modulators of the IL-1 Receptor St-Cyr D.J., Beauregard K., Bernard-Gauthier V., *$Lubell W.D.
18:00 01060 Enhancing Therapeutic Potentials of Nordihydroguaiaretic Acid (NDGA) through Synthesis and Metabolism Studies of novel Phenol and Catechol NDGA Analogues Asiamah I., Maloney K.A., *$Krol E.S.
18:00 01061 Second Generation Purine Inhibitors of Stat3 Show Greater Than 6-fold Increased Activity Over Previous Library Shahani V.M., Ball D.P., $Gunning P.T.
18:00 01062 Multivalent Salicylic Acid Based Small Molecule Inhibitors of Protein Tyrosine Phosphatases Ball D.P., Haftchenary S., Aubry I., Page B.D.G., Shahani V.M., Tremblay M., $Gunning P.T.
18:00 01063 Design and Synthesis of Glutathione Peroxidase Mimetics Press D.J., $Back T.G.
18:00 01064 Studies Related to Glutathione Peroxidase Mimetics McNeil N.M.R., Press D.J., *$Back T.G.
18:00 01065 Progress Toward the Synthesis of Labeled Derivatives of the Cystic Fibrosis Drug, Ivacaftor Elmallah S., *$Viirre R.D.
18:00 01066 Amines with Boron: Good for your Wood! Bowes E.G., Campbell-Verduyn L.S., Smash L.T., Vogels C.M., Decken A., Baerlocher F.J., Betsch M.P., *$Westcott S.A.
18:00 01067 Novel Capsaicin Derivatives for the Treatment of Cancer Patterson A.E., Bowes E.G., Fontaine F.-G., Culf A.S., Ramsaywack S., Decken A., *$Westcott S.A.
18:00 01068 Design and Synthesis of Novel Inhibitors of the Influenza A Virus Neuraminidase Jabari N., $Pinto B.M.
18:00 01069 Umbrella-rotaxanes : Towards New Vehicles for Anions and Drugs Transporters Richard-Daniel J., Chhun C., $Schmitzer A.R.
18:00 01070 Synthesis of an Inhibitor of Glutamate-1-Semialdehyde Aminomutase Nadeau A.K., *$Sorensen J.L.

OR6 - Applied Photochemistry in Health Research posters

18:00 01071 New Colored-substrates for Facile Determination of Activity and Biocatalytic Parameters of Chloroperoxidase $Najjar-Safari A., *Nazari K., Adhami F., Mahmoudi A.
18:00 01072 Optimising Two-photon Photodynamic Therapy in the Chicken CAM Model Probodh I., *$Cramb D.T.
18:00 01073 Synthesis of Photo-affinity Probes to Determine Site and Specificity of Inhibitor Binding in MRSA Bagha B.S., Jonadass J.P.S., *Kumar N.S., $Young R.N.
18:00 01074 Do all Fluorescent Proteins React with Singlet Oxygen? Gutierrez R., Valencia-Perez A.Z., *$Heyne B.

OR7 - Carbohydrate Chemistry and Glycobiology posters

18:00 01075 Anti-Bacterial Activity of UDP-Galactopyranose Mutase Inhibitors Borrelli S., Mohan S., *$Pinto B.M.
18:00 01076 Characterization of Carbohydrate Binding Domain of Clostridium diffcile Toxin A Zhang P., Eugenio L., Ng K.K.-S., *Ling C.-C.
18:00 01077 Easily Accessible Mannosides *Al-Mughaid H., Twibanire J.-d'.K., $Grindley T.B.
18:00 01078 Synthesis of Sugar Phosphates that are Putative Intermediates in Aminosugar Biosynthesis in Bacillus subtilis. Jagdhane R., Anjum S., *$Palmer D.R.
18:00 01079 Efficient Synthesis of a Novel a-Cyclodextrin-based Capsule Wang A.X., Li W.L., *Ling C.-C.
18:00 01080 Computational Study of Hydroxyproline Oligo-glycopeptides Naziga E.B., Schweizer F., *$Wetmore S.D.
18:00 01081 Progress Towards the Synthesis of the Chimeric Glycopeptide Corresponding to the Shigella flexneri Y O- Polysaccharide and its Peptide Mimic MDWNMHAA Challa V.R., Hossany R.B., *$Pinto B.M.
ORMacleod E1

Ligand Design (joint with IN4)

13:40 See IN4.

17:20 End of Session

ORMacleod D

Molecular Design of Optical, Photonic and Electronic Materials

13:40 Joint with MT and IN - See MT2.

17:40 End of Session

ORTELUS 105

Teaching Organic Chemistry (joint with CE3)

13:40 See CE3.

17:00 End of Session


Tuesday AM

OR3Macleod C

Symposium in Honour of Edward Piers

Organizer(s) - V. Snieckus
Chair(s) - V. Snieckus

08:10 Introductory Remarks

08:20 01269 The Discovery and Development of Phosphodiesterase-4 Inhibitors Friesen R.W.
09:00 01270 The Synthesis of Gigasol: A Natural Product Isolated from Angelica gigas that is Used in Korean Folk Medicine Gorobets E., *$Keay B.A.
09:40 01271 Synthetic Studies on Marine Polypropionates Becerril-Jiménez F., Zahedi M. M., Ward D.E.
10:00 Coffee Break
10:20 01272 Development of Practicle Syntheses for the Preparation of Novel Drug Targets Morton H.E.
11:00 01273 Palladium-Catalyzed Reactions Proceeding via b-Carboelimination of Tertiary Alcohols *$Orellana A., Rosa D., Chtchemelinine A., Nikolaev A., Schweinitz A.
11:20 01274 Reactivity of Oxa- and Azarhodacyclobutanes: On the Road to Novel Catalytic Transformations Dauth A., *$Love J.A.
11:40 01275 Greening Up Cross-Couplings Catalyzed by Copper & Palladium Using Tin and Related Organometallics *Lipshutz B.
12:20 End of Session

OR4Macleod B

Advances in Synthetic Methods

Organizer(s) - T. Back
Chair(s) - T. Back

08:10 Introductory Remarks

08:20 01276 Catalytic Nucleophilic Additions of Terminal Alkynes in Water *$Li C.-J.
09:00 01277 New Approaches to Aromatic Heterocycles using Heterogeneous Solvent-free Strategies *$Magolan J.
09:20 01278 Development of New Heterocyclic Systems via Geminal Acylation of Amino Acid-Based Oxazolidines Moulins J.R., $Burnell D.J.
09:40 01279 Carbon-Based Leaving Group Substitutions at sp3-Hybridized Benzylic Carbon Centers Mahoney S.J., Lou T., Bondarenko G., *$Fillion E.
10:00 Coffee Break
10:20 01280 Ring Contractions of N-Activated Lactams *$Spino C., Lessard J., Pichette S., Aubert-Nicol S., Winter D., Drouin A.
11:00 01281 Fluorine Transfer to Alkyl Radicals Rueda-Becerril M., Chatalova Sazepin C., Leung J.C.T., Okbinoglu T., Kennepohl P., Paquin J.-F., *$Sammis G.M.
11:20 01282 The Cyclization Chemistry Of Benzyl Alkynyl Sulfones *$Schwan A.L., Hossain M.S., Ho L.
11:40 01283 The Reactivity of Cyclopropane Hemi-malonates Emmett M.R., $Kerr M.A.
12:00 01284 Hydrogenative C-C Bond Formation for Syntheses of Homopropargylic Alcohols Geary L.M., $Krische M.J.
12:20 End of Session

OR8Macleod E1

General

Organizer(s) - T. Sutherland
Chair(s) - C. Smith

08:00 01285 Cobalt- and Nickel-Catalyzed Ester Hydrogenation. Dealklyation by Hydrogenolytic sp3 C-O Bond Activation Yu S., *$Stryker J.M.
08:20 01286 Boronic Acid Catalysis as a Mild and Versatile Strategy for Direct Carbo- and Hetero- Cyclizations of Free Allylic Alcohols Zheng H., Ghanbari S., Nakamura S., *$Hall D.G.
08:40 01287 From a-Boryl Aldehydes: An Adventure in the Reactivity of Amphoteric Molecules He Z., *$Yudin A. K.
09:00 01288 Towards a Formal Synthesis of Triptolide via a Gold-Catalyzed Cyclization Cascade Schwantje T., $Barriault L.
09:20 01289 Silyl Enol Ethers as Key Substrates in the Synthesis of 3-fluorofurans via Gold-Catalyzed 5-endo-dig Cycloisomerization *$Dembinski R., Li Y.
09:40 01290 Preparation of b-Boronyl-b-Aryl Enoates and their Subsequent Copper-Catalyzed Asymmetric Conjugate Reduction to Produce Chiral Secondary Alkylboronates Ding J., Lee J.C.H., *$Hall D.G.
10:00 Coffee Break
10:20 01291 Catalytic Enantioselective Allylboration of Propargylic Aldehydes Bhakta U., Graham E., *$Hall D.G.
10:40 01292 The Total Synthesis of Muamvatin Zahedi M.M., $Ward D.E.
11:00 01293 Studies Towards a Total Synthesis of (-)-Amphidinolide K Campbell N.E., $Sammis G.M.
11:20 01294 An Expedient Synthesis of Chiral Polysubstituted 1,4-Oxazepines *Bezanson M., $Moitessier N.
11:40 01295 Stereoselective Synthesis of Brevianamide E Zhao L., May J., Huang J., *$Perrin D.
12:00 01296 Tetrasubstituted Porphyrins Synthesized by Mechanochemistry $Hamilton T.D., Mackin P.
12:20 End of Session

ORMacleod D

Molecular Design of Optical, Photonic and Electronic Materials

08:00 Joint with MT and IN - See MT2.

12:20 End of Session


Tuesday PM

OR3Macleod C

Symposium in Honour of Edward Piers

Organizer(s) - V. Snieckus
Chair(s) - V. Snieckus

13:40 01510 New Samarium Diiodide Mediated Cascade Reactions to Heterocycles: A Short Route to Strychnine Reissig H.
14:20 01511 New Applications for Chlorohydrins in Natural Product Synthesis *$Britton R.A.
15:00 Break

15:20 01512 Function Oriented Synthesis of Marine Natural Product Pharmacophores Andersen R.J.
16:00 01513 Second Generation Hepatitis C Virus NS3 Protease Inhibitors with Improved Antiviral Profile Llinas-Brunet M.
16:20 End of Session

OR4Macleod B

Advances in Synthetic Methods

Organizer(s) - T. Back
Chair(s) - T. Back

13:40 01514 Approaches to Lysergic Acid Via Ammonium Ylide Rearrangement Dunbar C.R., $West F.G.
14:00 01515 Chemoenzymatic Approach to Diverse Analogues of Pancratistatin and Narciclasine Vshyvenko S., Scattolon J., *$Hudlicky T.
14:20 01516 Some Adventures in Synthesis: Natural Products and Methodology *Clive D.L.J.

Alfred Bader Award lecture:

15:00 01517 From Free-Radicals to Polypropionates Guindon Y.
15:40 Break

16:00 01518 Recent Advances in the Synthesis of Heterocycles from Cyclopropanes *$Kerr M.A.
16:40 Coffee Break
17:00 End of Session


Wednesday AM

OR4Macleod B

Advances in Synthetic Methods

Organizer(s) - T. Back
Chair(s) - T. Back

08:00 01807 Progress Toward the Total Synthesis of Morphine via a Tandem Oxy-cope/Claisen/Ene Reaction *Marcotte J., Lepack K., $Barriault L.
08:20 01808 New Bond-Forming Processes Initiated by Nazarov Electrocyclization *$West F.G.
09:00 01809 Highly Chemo- and Enantioselective Cross-Benzoin Reaction of Aliphatic Aldehydes with a-Ketoesters Thai K., Bilodeau F., *Gravel M.
09:20 01810 Biocatalytic Synthesis of Alklaloids and Explorations of New Annulation Methods *Hudlicky T.
10:00 Coffee Break
10:20 01811 A New Route to 2-alkenyl/alkylidenyl-3-tert-butyldiphenylsilylamines *$Yadav V.K., Narhe B.D., Hulikal V.
10:40 01812 Advances and Applications of Aqueous Wittig-type Olefination Reactions McLeod D., *$McNulty J.
11:00 01813 Boronic Acid Catalysis: A Mild and Versatile Approach for Direct Activation of Alcohols and Carboxylic Acids *$Hall D.G.

Boehringer Ingelheim (Canada) Research Excellence Award lecture:

11:40 01814 Harvest in the Natural Product Synthesis and Gold-Catalyzed Gardens Barriault L.
12:20 End of Session

OR7Macleod C

Carbohydrate Chemistry and Glycobiology (joint with BM)

Organizer(s) - C.C. Ling, C. Cairo
Chair(s) - C. Cairo, D. Palmer

08:00 01815 Regio- and Chemoselective O-Desilylations to Access Multisubstituted Cyclodextrins: The Magic of Diisobutylaluminium Hydride (DIBAL-H) Ghosh R., Ling C.C.
08:20 01816 The Effects of Hydroxypoline Glycosylation on the Stability of Collagen *$Schweizer F., Bommagani S., Murthy V.
08:40 01817 A Synergistic Docking, MD and QM/MM Investigation on the First Stage of the Catalytic Mechanism of LuxS Huang W.-J., Gherib R., *$Gauld J.W.
09:00 01818 Conformational Analysis of Portions of the Mycobacterial Cell Wall Galactan via NMR and Molecular Dynamics Richards M.R., *$Lowary T.L.
09:20 01819 A Novel Biosynthetic Pathway to Aminosugars in Bacillus spp *$Palmer D.R.J., Vetter N.D., Anjum S., Boisvert J., Jhagdane R., van Straaten K.E., Sanders D.A.R.
09:40 01820 Synthesis of Genetically-Encoded Glycopeptide Libraries Displayed on Phage *$Derda R., Ng S., Jafari M.R., Matochko W.
10:00 Coffee Break
R.U. Lemieux Award lecture:

10:20 01821 Look What You Started, Ray! NMR Methods for Probing Protein-ligand Interactions Pinto B.M.
11:00 01822 Hijacking of Metabolic Pathways to Generate Glycosyltransferase Inhbiitors that Act in Cells Gloster T.M., Zandberg W.F., Heinonen J.E., Shen D.L., Deng L., *$Vocadlo D.J.
11:20 01823 Protecting Group Free Synthesis of Glycosyl Phosphates Mediated by a Cu(II)-Oxazoline Complex Edgar L.J.G., *Dasgupta S., $Nitz M.
11:40 01824 Polyester Glycodendrimers and Dendronized Polymers as Potential Antiadhesion Drugs Against Urinary Tract Infections *$Grindley T.B., Twibanire J.K.
12:00 01825 Chemical Approaches to the Investigation of Protein-Membrane Binding Interactions Using Synthetic Lipid Probes *$Best M.D., Rowland M.M., Bostic H.E., Gong D., Smith M.D.
12:20 End of Session

OR8Macleod A1

General

Organizer(s) - T. Sutherland
Chair(s) - D. Press

08:00 01826 Organocatalysis of (-)-Complanine $Kamanos K.A.D, *Withey J.M.
08:20 01827 Synthesis of Anomeric and Non-Anomeric Spiroketals Related to Didemnaketal A *$Wulff J.E., Davy J.A., Moreau B.
08:40 01828 Synthesising Terminal Alkynes Using Canola Oil *Brown B.A., Smith A.D., $Veinot J.G.C.
09:00 01829 New Routes to Functional Silicones: The Design and Synthesis of Explicit 3-D Siloxane Macrostructures Grande J.B., $Brook M.A.
09:20 01830 Verdazyl Radicals in Organic Synthesis Bancerz M., $Georges M.K.
09:40 01831 Asymmetric 1,3-Dipolar Cycloaddition of Azomethine Imine made In Situ from Verdazyl Radical Youn B., $Georges M.K.
10:00 Coffee Break
10:20 01832 Supramolecular Induction of Chirality in a New Catalytic Biotin-functionnalized Imidazolium Salt Gauchot V., *Schmitzer A.R.
10:40 01833 Application of Ionic Liquids as an Efficient Catalyst to Synthesize of High-performance Diketopyrrolopyrrole Pigments *$Nourmohammadian F., Shamekhi S.
11:00 01834 Synthetic Studies on the ABC-Tricyclic Core of Manzamine B *Donahue J., $MaGee D.
11:20 01835 The Azide Captured Nazarov Reaction: Synthesis and Reactivity of the [3+3]-Cycloadducts Scadeng O., *$West F.G.
11:40 01836 The Oxidative Nazarov Reaction Kwon Y., *West F.G.
12:00 End of Session

ORTELUS 106

Radiopharmaceutical Chemistry (joint with BM3)

08:00 See BM3.

12:20 End of Session


Wednesday PM

OR4Macleod B

Advances in Synthetic Methods

Organizer(s) - T. Back
Chair(s) - T. Back

13:40 01959 Novel Stereoselective C-H Amination Reactions: A Green Perspective *$Lebel H., Trudel C., Mamani-Laparra L.
14:20 01960 Progress in the Palladium-Catalyzed Cross-Couplings Employing CO2 and SO2 Extrusions to Form Biaryls Forgione P.
14:40 01961 Revisiting the Use of Fluoride as a Leaving Group *Paquin J.-F.

Boehringer Ingelheim (Canada) Doctoral Research Award lecture:

15:00 01962 Development of Cross-Coupling and Cycloaddition Reactions Marcoux D.
15:40 Coffee Break
16:00 01963 A Surprising Ene-Type Reaction In An Isodicyclopentadiene Derivative Toward Taxinine Total Synthesis Joy S., Nakanishi W., Benson C.L., Mazzola Jr. R.D., Giese S., *West F.G.
16:20 01964 Synthetic Studies Towards MPC1001F: A Natural Product Containing a Triketopiperazine and a Dihydrooxepin Ring Bhattacharyya D., *Peng J., $Clive D.L.J.
16:40 01965 Enantioselective Preparation and Chemoselective Cross-Coupling of 1,1-Diboron Compounds Lee J.C.H., McDonald R., *$Hall D.G.
17:00 01966 An N-Heterocyclic Carbene/Lewis Acid Strategy for the Stereoselective Synthesis of Spirooxindole Lactones Dugal-Tessier J., O'Bryan E.A., Schroeder T.B.H., Cohen D.T., *$Scheidt K.A.
17:20 End of Session

OR7Macleod C

Carbohydrate Chemistry and Glycobiology (joint with BM)

Organizer(s) - C.C. Ling, C. Cairo
Chair(s) - M. Nitz, C.-C. Ling

13:40 01967 Synthesis of an Idopyranoside-containing Capsular Polysaccharide Repeating Unit from Campylobacter jejuni Hevey R., *$Ling C.-C.
14:00 01968 From Chemical Glycosylation to Expeditious Oligosaccharide Synthesis *$Demchenko A.V.
14:40 01969 Design and Synthesis of a New Class of Glycosylphosphate Isosteres Downey A.M., *Cairo C.W.
15:00 01970 Approaches to C-Glycosides for use in C-Glycopeptide and C-Glycolipid Synthesis *$Gagne M.
15:20 01971 Catalyst-controlled, Regioselective Protection and Glycosylation of Carbohydrate Derivatives *$Taylor M.S., Dimitrijevic E., Gouliaras C., Lee D.
15:40 Coffee Break
Bernard Belleau Award lecture:

16:00 01972 Protein Recognition of Bacterial Glycans Containing Furanose Residues Lowary T.L.
16:40 01973 N-glycosides with Uses from Protecting-Group-Free Glycosidations to Site-Specific Protein Modifications *Nitz M.
17:00 01974 Probing b-Phosphoglucomutase Using Monofluoromethylenephosphonates: Insight in Transition State Mimicry *$Jakeman D.L.
17:20 End of Session

ORTELUS 106

Radiopharmaceutical Chemistry (joint with BM3)

13:40 See BM3.

17:40 End of Session


Top of Conference Schedule

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